Vesamicol is an experimental drug, acting presynaptically by inhibiting acetylcholine (ACh) uptake and reducing its release.

[3H]vesamicol binding in human brain cholinergic deficiency disorders
Vesamicol analogues as sigma ligands : Molecular determinants of selectivity at the vesamicol receptor
[3H]vesamicol binding in brain: Autoradiographic distribution, pharmacology, and effects of cholinergic lesions
Linkage of the acetylcholine transporter-vesamicol receptor to proteoglycan in synaptic vesicles
Empty synaptic vesicles recycle and undergo exocytosis at vesamicol-treated motor nerve terminals
Mouse brain distribution of a carbon-11 labeled vesamicol derivative: presynaptic marker of cholinergic neurons.
A kinetic and allosteric model for the acetylcholine transporter-vesamicol receptor in synaptic vesicles.
Cloning and expression of the vesamicol binding protein from the marine ray Torpedo. Homology with the putative vesicular acetylchol...
Choline acetyltransferase activity and [3H]vesamicol binding in the temporal cortex of patients with Alzheimer's disease, Parkinson'...
Effects of Systemic Administration of 2-(4-Phenyl-Piperidino)-Cyclohexanol (Vesamicol) and an Organophosphate DDVP on the Cholinergi...